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INHIBITORS OF PI3K

Expression

Ubiquitous

Ubiquitous

Leukocytes

Leukocytes

Insulin signaling

Mutated in solid

tumours

Platelet activation

Neutrophil function

Insulin signaling

Mast cell activation

Innate immunity

Immune tracking

B and T cell activation

Fc receptor signaling

Idelalisib

Duvelisib

Copanlisib

TG-1202

a

b

g

d

Class I PI3K

Isoform